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SIMM · NJU
Assay
PGDB_AS002503
System: cell_based
Target: IKZF2
Cell line: 293GT
Assay context summary
Assay context
25 activity records
Assay family
% Degradation
System
cell_based
Readout
EC50
Target
IKZF2
E3
Not specified
Cell line
293GT
Detection target
protein_degradation
Activity compounds and values
Activity records
25 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
=
0.029
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A014227
PGDB_C008712
PGDB_AS002503
View
EC50
-
=
0.066
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A015188
PGDB_C008958
PGDB_AS002503
View
EC50
-
=
0.049
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A021323
PGDB_C008952
PGDB_AS002503
View
EC50
-
=
0.23
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A023498
PGDB_C008949
PGDB_AS002503
View
EC50
-
=
0.73
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A026226
PGDB_C008947
PGDB_AS002503
View
EC50
-
>
30
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A027782
PGDB_C008959
PGDB_AS002503
View
EC50
-
>
30
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A031756
PGDB_C008938
PGDB_AS002503
View
EC50
-
=
1.67
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A033452
PGDB_C008943
PGDB_AS002503
View
EC50
-
=
0.103
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A036942
PGDB_C008940
PGDB_AS002503
View
EC50
-
=
0.45
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A037577
PGDB_C008955
PGDB_AS002503
View
EC50
-
=
0.024
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A038931
PGDB_C008950
PGDB_AS002503
View
EC50
-
=
0.99
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A039393
PGDB_C008960
PGDB_AS002503
View
EC50
-
=
0.67
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A039733
PGDB_C008954
PGDB_AS002503
View
EC50
-
=
1.57
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A040251
PGDB_C008961
PGDB_AS002503
View
EC50
-
=
0.1
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A045454
PGDB_C008944
PGDB_AS002503
View
EC50
-
=
0.41
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A051965
PGDB_C008962
PGDB_AS002503
View
EC50
-
=
0.23
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A060545
PGDB_C008953
PGDB_AS002503
View
EC50
-
=
0.036
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A067761
PGDB_C008946
PGDB_AS002503
View
EC50
-
=
0.043
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A067771
PGDB_C008941
PGDB_AS002503
View
EC50
-
=
0.15
uM
-
—
IKZF2
-
293GT
KR20210031923A
PGDB_A068521
PGDB_C008951
PGDB_AS002503
View