PatGlueDB | Molecular Glue Patent Bioactivity Database

Assay context summary

Assay context

72 activity records

Assay family% Degradation

Systemcell_based

ReadoutDC50

TargetGSPT1

E3Not specified

Cell lineCAL-51

OrganismHomo sapiens

Technologyfluorescence

Activity compounds and values

Activity records

72 records

Metric	Control	Relation	Value	Unit	Concentration	Time	Target	E3	Cell line	Patent	Record ID	Compound	Assay	Details
DC50	-	>	300	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A007196	PGDB_C009979	PGDB_AS002523	View
DC50	-	<=	30	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A009177	PGDB_C009951	PGDB_AS002523	View
DC50	-	<=	30	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A012726	PGDB_C009915	PGDB_AS002523	View
DC50	-	=	30-300	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A013769	PGDB_C009909	PGDB_AS002523	View
DC50	-	<=	30	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A014594	PGDB_C009931	PGDB_AS002523	View
DC50	-	<=	30	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A014681	PGDB_C009922	PGDB_AS002523	View
DC50	-	=	30-300	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A015089	PGDB_C009928	PGDB_AS002523	View
DC50	-	=	30-300	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A015610	PGDB_C009949	PGDB_AS002523	View
DC50	-	=	30-300	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A016998	PGDB_C009912	PGDB_AS002523	View
DC50	-	<=	30	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A019030	PGDB_C009956	PGDB_AS002523	View
DC50	-	<=	30	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A020915	PGDB_C009935	PGDB_AS002523	View
DC50	-	=	30-300	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A025218	PGDB_C009948	PGDB_AS002523	View
DC50	-	<=	30	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A026338	PGDB_C009914	PGDB_AS002523	View
DC50	-	<=	30	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A028812	PGDB_C009958	PGDB_AS002523	View
DC50	-	<=	30	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A029396	PGDB_C009954	PGDB_AS002523	View
DC50	-	<=	30	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A030062	PGDB_C009913	PGDB_AS002523	View
DC50	-	<=	30	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A031237	PGDB_C009964	PGDB_AS002523	View
DC50	-	=	30-300	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A031351	PGDB_C009911	PGDB_AS002523	View
DC50	-	=	30-300	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A032727	PGDB_C009924	PGDB_AS002523	View
DC50	-	<=	30	nM	-	—	GSPT1	-	CAL-51	WO2022219407A1	PGDB_A033720	PGDB_C009942	PGDB_AS002523	View

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