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SIMM · NJU
Assay
PGDB_AS002575
System: cell_based
Target: CDK2
Cell line: HEK293
Assay context summary
Assay context
45 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
CDK2
E3
Not specified
Cell line
HEK293
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
45 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A007194
PGDB_C027513
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A008837
PGDB_C027499
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A010580
PGDB_C027547
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A011328
PGDB_C027461
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A012934
PGDB_C027500
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A013709
PGDB_C027535
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A014204
PGDB_C027478
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A020515
PGDB_C027550
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A025026
PGDB_C027512
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A025606
PGDB_C027528
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A027963
PGDB_C027505
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A028247
PGDB_C027484
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A029387
PGDB_C027501
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A030832
PGDB_C027508
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A032332
PGDB_C027538
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A033801
PGDB_C027453
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A034418
PGDB_C027546
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A036325
PGDB_C027541
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A037878
PGDB_C027540
PGDB_AS002575
View
Dmax
-
>
80
%
30 uM
24 h
-
-
HEK293
WO2024092039
PGDB_A042547
PGDB_C027510
PGDB_AS002575
View