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O=C1CCC(c2c(F)cc(N3CC(NC(=O)Nc4cc(F)c5c(c4)OCC54CC4)C3)cc2F)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 16 | nM | - | — | GSPT1 | - | ABC-1 | CN119264113A | PGDB_A016249 | PGDB_C000672 | PGDB_AS001474 | View | |
| DC50 | - | = | 46.7 | nM | - | — | GSPT1 | - | CAL-51 | CN119264113A | PGDB_A017738 | PGDB_C000672 | PGDB_AS001139 | View | |
| IC50 | - | = | 8.4 | nM | - | — | GSPT1 | - | CAL-51 | CN119264113A | PGDB_A044099 | PGDB_C000672 | PGDB_AS001498 | View | |
| IC50 | - | = | 0.5 | nM | - | — | GSPT1 | - | ABC-1 | CN119264113A | PGDB_A056672 | PGDB_C000672 | PGDB_AS002488 | View |