Assay
PGDB_AS001498
System: cell_basedCell line: CAL-51
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | > | 1000 | nM | - | — | GSPT1 | - | CAL-51 | CN119264113A | PGDB_A019641 | PGDB_C000675 | PGDB_AS001498 | View | |
| IC50 | - | = | 8.4 | nM | - | — | GSPT1 | - | CAL-51 | CN119264113A | PGDB_A044099 | PGDB_C000672 | PGDB_AS001498 | View | |
| IC50 | - | = | 68.9 | nM | - | — | GSPT1 | - | CAL-51 | CN119264113A | PGDB_A061884 | PGDB_C000671 | PGDB_AS001498 | View | |
| IC50 | - | = | 10 | nM | - | — | GSPT1 | - | CAL-51 | CN119264113A | PGDB_A064049 | PGDB_C000673 | PGDB_AS001498 | View | |
| IC50 | - | = | 24.6 | nM | - | — | GSPT1 | - | CAL-51 | CN119264113A | PGDB_A072217 | PGDB_C000674 | PGDB_AS001498 | View |