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Cc1nc2cccc(SCCCN3CCN(C(c4ccc(F)cc4)c4ccc(F)cc4)CC3)c2c(=O)n1C1CCC(=O)NC1=O| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 204 | nM | - | — | - | - | TMD8 | WO2023151635A1 | PGDB_A008872 | PGDB_C001157 | PGDB_AS000648 | View | |
| IC50 | - | = | 285.6 | nM | - | — | - | - | Daudi | WO2023151635A1 | PGDB_A017902 | PGDB_C001157 | PGDB_AS000279 | View | |
| IC50 | - | = | 275.8 | nM | - | — | - | - | MM.1R | WO2023151635A1 | PGDB_A062438 | PGDB_C001157 | PGDB_AS001111 | View | |
| IC50 | - | = | 489.7 | nM | - | — | - | - | Ramos | WO2023151635A1 | PGDB_A071975 | PGDB_C001157 | PGDB_AS002135 | View |