Assay
PGDB_AS001111
System: cell_basedCell line: MM.1R
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 12.7 | nM | - | — | - | - | MM.1R | WO2023151635A1 | PGDB_A009697 | PGDB_C001156 | PGDB_AS001111 | View | |
| IC50 | - | = | 32.8 | nM | - | — | - | - | MM.1R | WO2023151635A1 | PGDB_A015334 | PGDB_C001158 | PGDB_AS001111 | View | |
| IC50 | - | = | 9.8 | nM | - | — | - | - | MM.1R | WO2023151635A1 | PGDB_A020691 | PGDB_C001164 | PGDB_AS001111 | View | |
| IC50 | - | = | 464.4 | nM | - | — | - | - | MM.1R | WO2023151635A1 | PGDB_A041227 | PGDB_C008731 | PGDB_AS001111 | View | |
| IC50 | - | = | 352.3 | nM | - | — | - | - | MM.1R | WO2023151635A1 | PGDB_A053029 | PGDB_C001159 | PGDB_AS001111 | View | |
| IC50 | - | = | 204.3 | nM | - | — | - | - | MM.1R | WO2023151635A1 | PGDB_A061641 | PGDB_C001177 | PGDB_AS001111 | View | |
| IC50 | - | = | 275.8 | nM | - | — | - | - | MM.1R | WO2023151635A1 | PGDB_A062438 | PGDB_C001157 | PGDB_AS001111 | View |