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Compound
PGDB_C002283
3 activity records1 related patents
2D structure
COc1ccc2c(c1)nc([C@H]1CC[C@H](NC(=O)c3cc(CNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)ccn3)CC1)n2CCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | < | 100 | nM | - | — | GSPT1 | - | HEK293 | WO2023237116A1 | PGDB_A041120 | PGDB_C002283 | PGDB_AS002200 | View |
| GI50 | - | < | 100 | nM | - | — | GSPT1 | - | HL-60 | WO2023237116A1 | PGDB_A048323 | PGDB_C002283 | PGDB_AS001555 | View |
| GI50 | - | = | 0.93 | nM | - | — | GSPT1 | - | Toledo | WO2023237116A1 | PGDB_A056594 | PGDB_C002283 | PGDB_AS002036 | View |