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SIMM · NJU
Assay
PGDB_AS002200
System: cell_based
Target: GSPT1
Cell line: HEK293
Assay context summary
Assay context
86 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
GSPT1
E3
Not specified
Cell line
HEK293
Technology
luminescence
Activity compounds and values
Activity records
86 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A009125
PGDB_C002253
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A009352
PGDB_C002274
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A009563
PGDB_C002266
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A010038
PGDB_C002214
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A010570
PGDB_C002237
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A010862
PGDB_C002206
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A011994
PGDB_C002260
PGDB_AS002200
View
DC50
-
=
100-1000
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A012610
PGDB_C002245
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A014996
PGDB_C002220
PGDB_AS002200
View
DC50
-
=
100-1000
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A015122
PGDB_C002285
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A015482
PGDB_C021177
PGDB_AS002200
View
DC50
-
=
100-1000
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A015985
PGDB_C002222
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A016592
PGDB_C002256
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A018878
PGDB_C002265
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A020639
PGDB_C002213
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A020737
PGDB_C002279
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A020941
PGDB_C002267
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A023725
PGDB_C002268
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A024180
PGDB_C002289
PGDB_AS002200
View
DC50
-
<
100
nM
-
—
GSPT1
-
HEK293
WO2023237116A1
PGDB_A025317
PGDB_C002288
PGDB_AS002200
View