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O=C1CCC(N2Cc3cc(CN4CC5CCC(C4)N5C(=O)c4ccccc4-c4ccc(Cl)cc4)ccc3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | <= | 5 | nM | - | — | - | - | Mino | WO2024032689A1 | PGDB_A010071 | PGDB_C002512 | PGDB_AS001319 | View | |
| IC50 | - | = | 10-50 | nM | - | — | - | - | CCRF-CEM | WO2024032689A1 | PGDB_A015425 | PGDB_C002512 | PGDB_AS001396 | View | |
| IC50 | - | = | 10-50 | nM | - | — | - | - | MM.1S | WO2024032689A1 | PGDB_A027197 | PGDB_C002512 | PGDB_AS001703 | View | |
| IC50 | - | = | 0.44 | uM | - | — | CRBN | CRBN | - | WO2024032689A1 | PGDB_A041329 | PGDB_C002512 | PGDB_AS000095 | View |