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Compound
PGDB_C003559
6 activity records1 related patents
2D structure
Cc1ccc(-c2c(-c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)cnn2C)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | < | 25 | nM | - | — | CSNK1A1 | - | HEK293 | EP4584259A1 | PGDB_A016962 | PGDB_C003559 | PGDB_AS001103 | View |
| EC50 | - | < | 100 | nM | - | — | - | - | - | EP4584259A1 | PGDB_A018897 | PGDB_C003559 | PGDB_AS002128 | View |
| % Degradation | - | = | 0-25 | % | Concentration range: 10 uM | six hours | GSPT1 | - | HEK293 | EP4584259A1 | PGDB_A024037 | PGDB_C003559 | PGDB_AS001220 | View |
| DC50 | - | >= | 25 | nM | - | — | GSPT1 | - | HEK293 | EP4584259A1 | PGDB_A039444 | PGDB_C003559 | PGDB_AS001862 | View |
| % Degradation | - | = | 75-90 | % | - | - | - | - | - | EP4584259A1 | PGDB_A068665 | PGDB_C003559 | PGDB_AS001586 | View |
| % Degradation | - | = | 75-90 | % | Concentration range: 10 uM | six hours | CSNK1A1 | - | HEK293 | EP4584259A1 | PGDB_A071464 | PGDB_C003559 | PGDB_AS000108 | View |