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Compound
PGDB_C004061
4 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(-c4cc(-c5ccccc5)n(C(F)F)n4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | >= | 25 | nM | - | — | CSNK1A1 | - | HEK293 | EP4584259A1 | PGDB_A007178 | PGDB_C004061 | PGDB_AS001103 | View |
| % Degradation | - | = | 0-25 | % | Concentration range: 10 uM | six hours | GSPT1 | - | HEK293 | EP4584259A1 | PGDB_A025291 | PGDB_C004061 | PGDB_AS001220 | View |
| % Degradation | - | = | 75-90 | % | Concentration range: 10 uM | six hours | CSNK1A1 | - | HEK293 | EP4584259A1 | PGDB_A033191 | PGDB_C004061 | PGDB_AS000108 | View |
| DC50 | - | >= | 25 | nM | - | — | GSPT1 | - | HEK293 | EP4584259A1 | PGDB_A054011 | PGDB_C004061 | PGDB_AS001862 | View |