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Compound
PGDB_C004111
4 activity records1 related patents
2D structure
CN1CCN(C(=O)c2cccc(-c3c(-c4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)ncn3C)c2)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | < | 25 | nM | - | — | CSNK1A1 | - | HEK293 | EP4584259A1 | PGDB_A007071 | PGDB_C004111 | PGDB_AS001103 | View |
| % Degradation | - | = | 0-25 | % | Concentration range: 10 uM | six hours | GSPT1 | - | HEK293 | EP4584259A1 | PGDB_A030692 | PGDB_C004111 | PGDB_AS001220 | View |
| % Degradation | - | = | 90-100 | % | Concentration range: 10 uM | six hours | CSNK1A1 | - | HEK293 | EP4584259A1 | PGDB_A045723 | PGDB_C004111 | PGDB_AS000108 | View |
| DC50 | - | >= | 25 | nM | - | — | GSPT1 | - | HEK293 | EP4584259A1 | PGDB_A053588 | PGDB_C004111 | PGDB_AS001862 | View |