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O=C1CCC(N2C(=O)c3ccc(NCCC[C@H]4C[C@@H](n5cc(-c6cnc7ccc(C8CCOCC8)cc7n6)c(C(F)(F)F)n5)C4)cc3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 10 | nM | - | — | - | - | MV-4-11 | WO2022073469A1 | PGDB_A008129 | PGDB_C004998 | PGDB_AS002199 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | MOLM-13 | WO2022073469A1 | PGDB_A035438 | PGDB_C004998 | PGDB_AS000571 | View | |
| IC50 | - | < | 10 | nM | - | — | GSPT1 | - | MOLM-13 | WO2022073469A1 | PGDB_A063283 | PGDB_C004998 | PGDB_AS000952 | View | |
| IC50 | - | < | 10 | nM | - | — | - | - | MV-4-11 | WO2022073469A1 | PGDB_A067634 | PGDB_C004998 | PGDB_AS000609 | View |