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O=C1CCC(N2C(=O)c3ccc(NC[C@H]4C[C@H](n5cc(-c6cc7cc[nH]c7cn6)c(C6CC6)n5)C4)cc3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 100-1000 | nM | - | — | - | - | MV-4-11 | WO2022073469A1 | PGDB_A007236 | PGDB_C005157 | PGDB_AS000609 | View | |
| IC50 | - | = | 10-100 | nM | - | — | - | - | MV-4-11 | WO2022073469A1 | PGDB_A011276 | PGDB_C005157 | PGDB_AS002199 | View | |
| IC50 | - | = | 10-100 | nM | - | — | GSPT1 | - | MOLM-13 | WO2022073469A1 | PGDB_A014908 | PGDB_C005157 | PGDB_AS000952 | View | |
| IC50 | - | >= | 1 | uM | - | — | GSPT1 | - | MOLM-13 | WO2022073469A1 | PGDB_A059406 | PGDB_C005157 | PGDB_AS000571 | View |