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Compound
PGDB_C005417
3 activity records1 related patents
2D structure
CCn1ncc(C(F)(F)F)c1-c1ccc(F)c(NC(=O)OCc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Potency ratio | Ref1 | = | 2-10 | fold | - | — | - | - | MDA-MB-468 | WO2025026218A1 | PGDB_A012414 | PGDB_C005417 | PGDB_AS001889 | View |
| Potency ratio | Ref1 | = | 1.3-2 | fold | - | — | - | - | NCI-H1155 | WO2025026218A1 | PGDB_A039915 | PGDB_C005417 | PGDB_AS001532 | View |
| % Inhibition | - | = | 52.6 | % | Concentration series: 3 uM, 5 uM, 10 uM | 5 min | KCNH2 | - | HEK293 | WO2025026218A1 | PGDB_A042813 | PGDB_C005417 | PGDB_AS000603 | View |