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Compound
PGDB_C006889
4 activity records1 related patents
2D structure
O=C(O)c1ccc2c(c1)OCCC(c1ccc(Cl)cc1Cl)=C2c1ccc(CC2CCN(CCCF)C2)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 5.4 | nM | - | — | ESR1 | - | MCF-7 | CN118984820A | PGDB_A014290 | PGDB_C006889 | PGDB_AS000996 | View |
| IC50 | - | = | 6.2 | nM | - | — | ESR1 | - | MCF-7 | CN118984820A | PGDB_A026580 | PGDB_C006889 | PGDB_AS000996 | View |
| % Degradation | - | = | 63 | % | 0.3 uM | 4 h | ESR1 | - | MCF-7 | CN118984820A | PGDB_A033006 | PGDB_C006889 | PGDB_AS001441 | View |
| % Degradation | - | = | 80 | % | 0.3 uM | 4 h | ESR1 | - | MCF-7 | CN118984820A | PGDB_A053582 | PGDB_C006889 | PGDB_AS001441 | View |