Assay

PGDB_AS000996

System: cell_basedTarget: ESR1Cell line: MCF-7
Assay context summary

Assay context

44 activity records
Assay family% Degradation
Systemcell_based
ReadoutIC50
TargetESR1
E3Not specified
Cell lineMCF-7
Activity compounds and values

Activity records

44 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C006912
IC50-=0.8nM-—ESR1-MCF-7CN118984820APGDB_A008714PGDB_C006912PGDB_AS000996View
2D structure for PGDB_C006920
IC50-=1.3nM-—ESR1-MCF-7CN118984820APGDB_A012432PGDB_C006920PGDB_AS000996View
2D structure for PGDB_C006901
IC50-=0.8nM-—ESR1-MCF-7CN118984820APGDB_A012912PGDB_C006901PGDB_AS000996View
2D structure for PGDB_C006920
IC50-=78.8nM-—ESR1-MCF-7CN118984820APGDB_A013992PGDB_C006920PGDB_AS000996View
2D structure for PGDB_C006914
IC50-=0.8nM-—ESR1-MCF-7CN118984820APGDB_A014181PGDB_C006914PGDB_AS000996View
2D structure for PGDB_C006889
IC50-=5.4nM-—ESR1-MCF-7CN118984820APGDB_A014290PGDB_C006889PGDB_AS000996View
2D structure for PGDB_C006913
IC50-=0.9nM-—ESR1-MCF-7CN118984820APGDB_A015732PGDB_C006913PGDB_AS000996View
2D structure for PGDB_C006886
IC50-=1.5nM-—ESR1-MCF-7CN118984820APGDB_A016145PGDB_C006886PGDB_AS000996View
2D structure for PGDB_C006922
IC50-=1.2nM-—ESR1-MCF-7CN118984820APGDB_A017455PGDB_C006922PGDB_AS000996View
2D structure for PGDB_C006919
IC50-=1.6nM-—ESR1-MCF-7CN118984820APGDB_A017584PGDB_C006919PGDB_AS000996View
2D structure for PGDB_C006918
IC50-=2nM-—ESR1-MCF-7CN118984820APGDB_A019931PGDB_C006918PGDB_AS000996View
2D structure for PGDB_C006891
IC50-=1.4nM-—ESR1-MCF-7CN118984820APGDB_A021332PGDB_C006891PGDB_AS000996View
2D structure for PGDB_C006906
IC50-=0.9nM-—ESR1-MCF-7CN118984820APGDB_A021898PGDB_C006906PGDB_AS000996View
2D structure for PGDB_C006892
IC50-=0.3nM-—ESR1-MCF-7CN118984820APGDB_A023258PGDB_C006892PGDB_AS000996View
2D structure for PGDB_C006908
IC50-=1.3nM-—ESR1-MCF-7CN118984820APGDB_A026296PGDB_C006908PGDB_AS000996View
2D structure for PGDB_C006889
IC50-=6.2nM-—ESR1-MCF-7CN118984820APGDB_A026580PGDB_C006889PGDB_AS000996View
2D structure for PGDB_C006899
IC50-=0.7nM-—ESR1-MCF-7CN118984820APGDB_A027282PGDB_C006899PGDB_AS000996View
2D structure for PGDB_C006895
IC50-=35nM-—ESR1-MCF-7CN118984820APGDB_A030820PGDB_C006895PGDB_AS000996View
2D structure for PGDB_C006883
IC50-=0.5nM-—ESR1-MCF-7CN118984820APGDB_A036753PGDB_C006883PGDB_AS000996View
2D structure for PGDB_C006903
IC50-=1.4nM-—ESR1-MCF-7CN118984820APGDB_A040265PGDB_C006903PGDB_AS000996View
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