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Compound
PGDB_C007551
6 activity records1 related patents
2D structure
N#Cc1ccc(N2CCN(Cc3ccc(Cc4ccc5c6c(cc(F)cc46)C(=O)N5C4CCC(=O)NC4=O)cc3)CC2)c(F)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.04 | nM | - | — | - | - | MM.1S | EP4393915A1 | PGDB_A021215 | PGDB_C007551 | PGDB_AS001514 | View |
| DC50 | - | = | 0.032 | uM | - | — | SALL4 | - | HT-1080 | EP4393915A1 | PGDB_A024504 | PGDB_C007551 | PGDB_AS000384 | View |
| DC50 | - | = | 0.074 | nM | - | — | IKZF1 | - | HT-1080 | EP4393915A1 | PGDB_A027666 | PGDB_C007551 | PGDB_AS001653 | View |
| Ymin | - | = | 4 | % | Concentration context: Y min : (%) | 120 h | - | - | MM.1S | EP4393915A1 | PGDB_A040043 | PGDB_C007551 | PGDB_AS002328 | View |
| Dmax | - | = | 91.6 | % | Concentration context: HiBiT IKZF1:_D max (%) | 20 h | IKZF1 | - | HT-1080 | EP4393915A1 | PGDB_A043916 | PGDB_C007551 | PGDB_AS001371 | View |
| Dmax | - | = | 58.1 | % | Concentration context: HiBiT SALL4:_D max (%) | 20 h | SALL4 | - | HT-1080 | EP4393915A1 | PGDB_A076082 | PGDB_C007551 | PGDB_AS001879 | View |