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Compound
PGDB_C007555
4 activity records1 related patents
2D structure
O=C1CCC(N2C(=O)c3cc(F)cc4c(Cc5ccc(CN6CCC(N7CCOCC7)CC6)cc5F)ccc2c34)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 2.19 | nM | - | — | IKZF1 | - | HT-1080 | EP4393915A1 | PGDB_A019854 | PGDB_C007555 | PGDB_AS001653 | View |
| Dmax | - | = | 33.9 | % | Concentration context: HiBiT SALL4:_D max (%) | 20 h | SALL4 | - | HT-1080 | EP4393915A1 | PGDB_A037346 | PGDB_C007555 | PGDB_AS001879 | View |
| Dmax | - | = | 66.2 | % | Concentration context: HiBiT IKZF1:_D max (%) | 20 h | IKZF1 | - | HT-1080 | EP4393915A1 | PGDB_A041155 | PGDB_C007555 | PGDB_AS001371 | View |
| DC50 | - | > | 10 | uM | - | — | SALL4 | - | HT-1080 | EP4393915A1 | PGDB_A056515 | PGDB_C007555 | PGDB_AS000384 | View |