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Compound
PGDB_C008439
4 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(C[C@H]4CCCC[C@@H]4NCc4cccnc4C(F)(F)F)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 75 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A012798 | PGDB_C008439 | PGDB_AS000211 | View |
| Dmax | - | = | 34 | % | - | 24 h | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A013504 | PGDB_C008439 | PGDB_AS000216 | View |
| EC50 | - | = | 0.046 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A033319 | PGDB_C008439 | PGDB_AS001535 | View |
| EC50 | - | = | 0.206 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A047702 | PGDB_C008439 | PGDB_AS002086 | View |