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SIMM · NJU
Assay
PGDB_AS002086
System: cell_based
Target: IKZF1
Cell line: HEK293
Assay context summary
Assay context
389 activity records
Assay family
% Degradation
System
cell_based
Readout
EC50
Target
IKZF1
E3
Not specified
Cell line
HEK293
Organism
Homo sapiens
Technology
luminescence
Detection target
protein_degradation
Activity compounds and values
Activity records
389 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
=
0.114
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A007014
PGDB_C008689
PGDB_AS002086
View
EC50
-
=
0.261
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A007279
PGDB_C008416
PGDB_AS002086
View
EC50
-
=
0.072
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A007349
PGDB_C008536
PGDB_AS002086
View
EC50
-
=
0.03
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A007791
PGDB_C008580
PGDB_AS002086
View
EC50
-
=
0.066
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A008131
PGDB_C008575
PGDB_AS002086
View
EC50
-
=
0.076
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A008366
PGDB_C008622
PGDB_AS002086
View
EC50
-
>
1
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A008782
PGDB_C008428
PGDB_AS002086
View
EC50
-
=
0.243
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A008833
PGDB_C008650
PGDB_AS002086
View
EC50
-
>
1
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A008937
PGDB_C008576
PGDB_AS002086
View
EC50
-
=
0.105
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A008951
PGDB_C008612
PGDB_AS002086
View
EC50
-
>
1
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A009044
PGDB_C008726
PGDB_AS002086
View
EC50
-
=
0.242
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A009383
PGDB_C008483
PGDB_AS002086
View
EC50
-
=
0.081
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A009457
PGDB_C008726
PGDB_AS002086
View
EC50
-
=
0.076
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A009550
PGDB_C008578
PGDB_AS002086
View
EC50
-
>
1
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A009764
PGDB_C008446
PGDB_AS002086
View
EC50
-
=
0.21
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A009783
PGDB_C008664
PGDB_AS002086
View
EC50
-
=
0.077
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A009974
PGDB_C008543
PGDB_AS002086
View
EC50
-
>
1
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A010003
PGDB_C008654
PGDB_AS002086
View
EC50
-
>
1
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A010070
PGDB_C008726
PGDB_AS002086
View
EC50
-
=
0.013
uM
-
—
IKZF1
-
HEK293
JP2026020265A
PGDB_A010156
PGDB_C008665
PGDB_AS002086
View