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CC(C)OC1CCC(N[C@H]2CCCC[C@@H]2Cc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.077 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A009974 | PGDB_C008543 | PGDB_AS002086 | View | |
| Dmax | - | = | 36 | % | - | 24 h | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A011321 | PGDB_C008543 | PGDB_AS000216 | View | |
| Dmax | - | = | 97 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A013858 | PGDB_C008543 | PGDB_AS000211 | View | |
| EC50 | - | = | 0.003 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A036494 | PGDB_C008543 | PGDB_AS001535 | View | |
| EC50 | - | = | 0.246 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A037042 | PGDB_C008543 | PGDB_AS002086 | View | |
| EC50 | - | = | 0.002 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A039081 | PGDB_C008543 | PGDB_AS001535 | View | |
| Dmax | - | = | 39 | % | - | 24 h | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A040650 | PGDB_C008543 | PGDB_AS000216 | View | |
| Dmax | - | = | 97 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A059612 | PGDB_C008543 | PGDB_AS000211 | View |