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CCC(C)N[C@H]1CCCC[C@@H]1Cc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 96 | % | - | 24 h | IKZF2 | - | - | JP2026020265A | PGDB_A007785 | PGDB_C008550 | PGDB_AS002581 | View | |
| Dmax | - | = | 98 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A009681 | PGDB_C008550 | PGDB_AS000211 | View | |
| EC50 | - | > | 1 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A015649 | PGDB_C008550 | PGDB_AS002086 | View | |
| EC50 | - | > | 1 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A046585 | PGDB_C008550 | PGDB_AS002086 | View | |
| EC50 | - | > | 1 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A050717 | PGDB_C008550 | PGDB_AS002086 | View | |
| EC50 | - | = | 0.002 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A052867 | PGDB_C008550 | PGDB_AS001535 | View | |
| Dmax | - | = | 97 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A060333 | PGDB_C008550 | PGDB_AS000211 | View | |
| EC50 | - | = | 0.002 | uM | - | — | IKZF2 | - | - | JP2026020265A | PGDB_A062980 | PGDB_C008550 | PGDB_AS001524 | View | |
| EC50 | - | = | 0.004 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A067284 | PGDB_C008550 | PGDB_AS001535 | View | |
| Dmax | - | = | 96 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A075702 | PGDB_C008550 | PGDB_AS000211 | View | |
| EC50 | - | = | 0.003 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A076055 | PGDB_C008550 | PGDB_AS001535 | View |