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COC1CCC(N[C@H]2CCCC[C@@H]2Cc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 98 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A009716 | PGDB_C008627 | PGDB_AS000211 | View | |
| EC50 | - | = | 0.114 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A011818 | PGDB_C008627 | PGDB_AS002086 | View | |
| Dmax | - | = | 37 | % | - | 24 h | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A039750 | PGDB_C008627 | PGDB_AS000216 | View | |
| Dmax | - | = | 37 | % | - | 24 h | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A044176 | PGDB_C008627 | PGDB_AS000216 | View | |
| EC50 | - | = | 0.004 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A047145 | PGDB_C008627 | PGDB_AS001535 | View | |
| Dmax | - | = | 98 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A051600 | PGDB_C008627 | PGDB_AS000211 | View | |
| Dmax | - | = | 95 | % | - | 24 h | IKZF2 | - | - | JP2026020265A | PGDB_A053750 | PGDB_C008627 | PGDB_AS002581 | View | |
| EC50 | - | = | 0.002 | uM | - | — | IKZF2 | - | - | JP2026020265A | PGDB_A056626 | PGDB_C008627 | PGDB_AS001524 | View | |
| EC50 | - | = | 0.003 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A059482 | PGDB_C008627 | PGDB_AS001535 | View | |
| EC50 | - | = | 0.125 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A075533 | PGDB_C008627 | PGDB_AS002086 | View |