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COC1(C)CCC(N[C@H]2CCCO[C@@H]2Cc2ccc3c(c2F)CN(C2CCC(=O)NC2=O)C3=O)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.243 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A008833 | PGDB_C008650 | PGDB_AS002086 | View | |
| Dmax | - | = | 95 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A026946 | PGDB_C008650 | PGDB_AS000211 | View | |
| EC50 | - | = | 0.006 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A041368 | PGDB_C008650 | PGDB_AS001535 | View | |
| EC50 | - | > | 1 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A046527 | PGDB_C008650 | PGDB_AS002086 | View | |
| Dmax | - | = | 33 | % | - | 24 h | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A050043 | PGDB_C008650 | PGDB_AS000216 | View | |
| Dmax | - | = | 94 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A063384 | PGDB_C008650 | PGDB_AS000211 | View | |
| EC50 | - | = | 0.007 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A064924 | PGDB_C008650 | PGDB_AS001535 | View | |
| EC50 | - | > | 10 | uM | - | — | SALL4 | - | HEK293 | JP2026020265A | PGDB_A066367 | PGDB_C008650 | PGDB_AS001573 | View |