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Compound
PGDB_C008659
8 activity records1 related patents
2D structure
O=C1CC[C@H](N2Cc3cc(C[C@H]4CCCC[C@@H]4NC4CCC(F)(F)CC4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.002 | uM | - | — | IKZF2 | - | - | JP2026020265A | PGDB_A023918 | PGDB_C008659 | PGDB_AS001524 | View |
| EC50 | - | > | 10 | uM | - | — | SALL4 | - | HEK293 | JP2026020265A | PGDB_A025838 | PGDB_C008659 | PGDB_AS001573 | View |
| Dmax | - | = | 62 | % | - | 24 h | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A043739 | PGDB_C008659 | PGDB_AS000216 | View |
| % Degradation | - | = | 0.63 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A044218 | PGDB_C008659 | PGDB_AS000906 | View |
| EC50 | - | = | 0.022 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A048421 | PGDB_C008659 | PGDB_AS002086 | View |
| Dmax | - | = | 94 | % | - | 24 h | IKZF2 | - | - | JP2026020265A | PGDB_A050553 | PGDB_C008659 | PGDB_AS002581 | View |
| Dmax | - | = | 98 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A055379 | PGDB_C008659 | PGDB_AS000211 | View |
| EC50 | - | = | 0.001 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A071215 | PGDB_C008659 | PGDB_AS001535 | View |