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Compound
PGDB_C008690
9 activity records1 related patents
2D structure
O=C1CCC(N2Cc3c(ccc(C[C@H]4OCCC[C@@H]4NC4CCC5(CC4)CC5(F)F)c3F)C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 43 | % | - | 24 h | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A013624 | PGDB_C008690 | PGDB_AS000216 | View |
| Dmax | - | = | 96 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A016551 | PGDB_C008690 | PGDB_AS000211 | View |
| EC50 | - | > | 10 | uM | - | — | SALL4 | - | HEK293 | JP2026020265A | PGDB_A031862 | PGDB_C008690 | PGDB_AS001573 | View |
| EC50 | - | = | 0.122 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A033808 | PGDB_C008690 | PGDB_AS002086 | View |
| Dmax | - | = | 95 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A036791 | PGDB_C008690 | PGDB_AS000211 | View |
| EC50 | - | = | 0.003 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A037218 | PGDB_C008690 | PGDB_AS001535 | View |
| EC50 | - | = | 0.003 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A040007 | PGDB_C008690 | PGDB_AS001535 | View |
| Dmax | - | = | 37 | % | - | 24 h | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A067490 | PGDB_C008690 | PGDB_AS000216 | View |
| EC50 | - | = | 0.045 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A074319 | PGDB_C008690 | PGDB_AS002086 | View |