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O=C1CCC(N2Cc3cc(C[C@H]4OCCC[C@@H]4NC4CCC(F)CC4)ccc3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | > | 10 | uM | - | — | SALL4 | - | HEK293 | JP2026020265A | PGDB_A007008 | PGDB_C008691 | PGDB_AS001573 | View | |
| EC50 | - | = | 0.017 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A009586 | PGDB_C008691 | PGDB_AS001535 | View | |
| EC50 | - | = | 0.015 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A012176 | PGDB_C008691 | PGDB_AS001535 | View | |
| EC50 | - | > | 10 | uM | - | — | SALL4 | - | HEK293 | JP2026020265A | PGDB_A012894 | PGDB_C008691 | PGDB_AS001573 | View | |
| EC50 | - | > | 1 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A034402 | PGDB_C008691 | PGDB_AS002086 | View | |
| EC50 | - | > | 1 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A039033 | PGDB_C008691 | PGDB_AS002086 | View | |
| Dmax | - | = | 87 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A046675 | PGDB_C008691 | PGDB_AS000211 | View | |
| Dmax | - | = | 85 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A061973 | PGDB_C008691 | PGDB_AS000211 | View |