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O=C1CC[C@H](N2Cc3c(ccc(C[C@H]4OCCC[C@@H]4N[C@H]4CC[C@@H](F)CC4)c3F)C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | > | 10 | uM | - | — | SALL4 | - | HEK293 | JP2026020265A | PGDB_A027381 | PGDB_C008693 | PGDB_AS001573 | View | |
| EC50 | - | > | 1 | uM | - | — | IKZF1 | - | HEK293 | JP2026020265A | PGDB_A035255 | PGDB_C008693 | PGDB_AS002086 | View | |
| Dmax | - | = | 97 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A038382 | PGDB_C008693 | PGDB_AS000211 | View | |
| % Degradation | - | = | 0.38 | % | - | 24 h | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A073111 | PGDB_C008693 | PGDB_AS000906 | View | |
| EC50 | - | = | 0.005 | uM | - | — | IKZF2 | - | HEK293 | JP2026020265A | PGDB_A074591 | PGDB_C008693 | PGDB_AS001535 | View |