Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C009077
3 activity records1 related patents
2D structure
O=C1CCC(N2Cc3c(CCCOCCOCCOCCCc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)cccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Kd | - | = | 11.15 | uM | - | — | CRBN | CRBN | - | US20220362229A1 | PGDB_A011461 | PGDB_C009077 | PGDB_AS002291 | View |
| % Inhibition | - | = | 76.25 | % | 200 uM | - | - | - | - | US20220362229A1 | PGDB_A041336 | PGDB_C009077 | PGDB_AS001773 | View |
| % Degradation | - | = | 12.45 | % | Concentration series: 10 nM, 10 uM | - | CRBN | CRBN | - | US20220362229A1 | PGDB_A052657 | PGDB_C009077 | PGDB_AS002247 | View |