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Compound
PGDB_C009085
3 activity records1 related patents
2D structure
O=C(/C=C/c1cccc2c1CN(C1CCC(=O)NC1=O)C2=O)NCCOCCOCCOCCNC(=O)/C=C/c1cccc2c1CN(C1CCC(=O)NC1=O)C2=OCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Kd | - | = | 8.21 | uM | - | — | CRBN | CRBN | - | US20220362229A1 | PGDB_A021359 | PGDB_C009085 | PGDB_AS002291 | View |
| % Inhibition | - | = | 83.88 | % | 200 uM | - | - | - | - | US20220362229A1 | PGDB_A022522 | PGDB_C009085 | PGDB_AS001773 | View |
| % Degradation | - | = | 59.08 | % | Concentration series: 10 nM, 10 uM | - | CRBN | CRBN | - | US20220362229A1 | PGDB_A037499 | PGDB_C009085 | PGDB_AS002247 | View |