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Compound
PGDB_C009088
3 activity records1 related patents
2D structure
O=C1CCC(N2Cc3c(NC(=O)CCCC(=O)Nc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)cccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Kd | - | = | 23.64 | uM | - | — | CRBN | CRBN | - | US20220362229A1 | PGDB_A013161 | PGDB_C009088 | PGDB_AS002291 | View |
| % Inhibition | - | = | 83.6 | % | 200 uM | - | - | - | - | US20220362229A1 | PGDB_A043566 | PGDB_C009088 | PGDB_AS001773 | View |
| % Degradation | - | = | 2.97 | % | Concentration series: 10 nM, 10 uM | - | CRBN | CRBN | - | US20220362229A1 | PGDB_A065291 | PGDB_C009088 | PGDB_AS002247 | View |