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COc1cc(N2CCC(N(C)Cc3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2S(C)(=O)=O)n1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 5000-10000 | nM | - | — | ALK | - | Mino | CN116239566A | PGDB_A023058 | PGDB_C019609 | PGDB_AS002386 | View | |
| IC50 | - | = | 100-500 | nM | - | — | ALK | - | MDA-MB-231 | CN116239566A | PGDB_A033030 | PGDB_C019609 | PGDB_AS000594 | View | |
| IC50 | - | < | 50 | nM | - | — | ALK | - | SR | CN116239566A | PGDB_A047558 | PGDB_C019609 | PGDB_AS001815 | View | |
| IC50 | - | = | 100-500 | nM | - | — | ALK | - | HCC827 | CN116239566A | PGDB_A060230 | PGDB_C019609 | PGDB_AS000527 | View | |
| IC50 | - | = | 100-500 | nM | - | — | ALK | - | PC-9 | CN116239566A | PGDB_A064698 | PGDB_C019609 | PGDB_AS000139 | View |