Assay
PGDB_AS002386
System: cell_basedCell line: Mino
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | Mino | CN116239566A | PGDB_A014591 | PGDB_C025913 | PGDB_AS002386 | View | |
| IC50 | - | = | 5000-10000 | nM | - | — | ALK | - | Mino | CN116239566A | PGDB_A023058 | PGDB_C019609 | PGDB_AS002386 | View | |
| IC50 | - | = | 100-500 | nM | - | — | ALK | - | Mino | CN116239566A | PGDB_A027277 | PGDB_C019613 | PGDB_AS002386 | View | |
| IC50 | - | = | 50-100 | nM | - | — | ALK | - | Mino | CN116239566A | PGDB_A036518 | PGDB_C025915 | PGDB_AS002386 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | Mino | CN116239566A | PGDB_A045574 | PGDB_C025912 | PGDB_AS002386 | View | |
| IC50 | - | = | 50-100 | nM | - | — | ALK | - | Mino | CN116239566A | PGDB_A048062 | PGDB_C025915 | PGDB_AS002386 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | ALK | - | Mino | CN116239566A | PGDB_A055974 | PGDB_C016074 | PGDB_AS002386 | View |