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Cc1cc(Nc2ncc(Cl)c(Nc3ccccc3S(=O)(=O)C(C)(C)C)n2)c(OC(C)C)cc1N1CCC(N(C)Cc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1000-5000 | nM | - | — | ALK | - | NCI-H1975 | CN116239566A | PGDB_A034155 | PGDB_C019611 | PGDB_AS002181 | View | |
| IC50 | - | < | 50 | nM | - | — | ALK | - | SR | CN116239566A | PGDB_A038067 | PGDB_C019611 | PGDB_AS001815 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | PC-9 | CN116239566A | PGDB_A038469 | PGDB_C019611 | PGDB_AS000139 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | MDA-MB-231 | CN116239566A | PGDB_A040009 | PGDB_C019611 | PGDB_AS000594 | View |