Assay
PGDB_AS002181
System: cell_basedCell line: NCI-H1975
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | ALK | - | NCI-H1975 | CN116239566A | PGDB_A022029 | PGDB_C016074 | PGDB_AS002181 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | ALK | - | NCI-H1975 | CN116239566A | PGDB_A034155 | PGDB_C019611 | PGDB_AS002181 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | NCI-H1975 | CN116239566A | PGDB_A039121 | PGDB_C025912 | PGDB_AS002181 | View | |
| IC50 | - | = | 50-100 | nM | - | — | ALK | - | NCI-H1975 | CN116239566A | PGDB_A040903 | PGDB_C019610 | PGDB_AS002181 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | ALK | - | NCI-H1975 | CN116239566A | PGDB_A073401 | PGDB_C025907 | PGDB_AS002181 | View | |
| IC50 | - | = | 50-100 | nM | - | — | ALK | - | NCI-H1975 | CN116239566A | PGDB_A073514 | PGDB_C019613 | PGDB_AS002181 | View |