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CNC(=O)c1ccccc1Nc1cc(Nc2ccc(N3CCC(N(C)Cc4ccc5c(c4F)CN(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1C(F)(F)F| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | SR | CN116239566A | PGDB_A031059 | PGDB_C019619 | PGDB_AS001780 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | SW620 | CN116239566A | PGDB_A044522 | PGDB_C019619 | PGDB_AS001904 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | PTK2 | - | PC-9 | CN116239566A | PGDB_A053650 | PGDB_C019619 | PGDB_AS001387 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | SW620 | CN116239566A | PGDB_A062432 | PGDB_C019619 | PGDB_AS001904 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | PTK2 | - | Mino | CN116239566A | PGDB_A070619 | PGDB_C019619 | PGDB_AS000370 | View | |
| IC50 | - | = | 50-100 | nM | - | — | PTK2 | - | VCaP | CN116239566A | PGDB_A077543 | PGDB_C019619 | PGDB_AS000495 | View |