Assay
PGDB_AS000370
System: cell_basedCell line: Mino
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | Mino | CN116239566A | PGDB_A007953 | PGDB_C025942 | PGDB_AS000370 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | Mino | CN116239566A | PGDB_A010887 | PGDB_C025941 | PGDB_AS000370 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | Mino | CN116239566A | PGDB_A011349 | PGDB_C025943 | PGDB_AS000370 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | Mino | CN116239566A | PGDB_A012143 | PGDB_C025944 | PGDB_AS000370 | View | |
| IC50 | - | = | 50-100 | nM | - | — | PTK2 | - | Mino | CN116239566A | PGDB_A028252 | PGDB_C025949 | PGDB_AS000370 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | Mino | CN116239566A | PGDB_A049008 | PGDB_C025940 | PGDB_AS000370 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | PTK2 | - | Mino | CN116239566A | PGDB_A055298 | PGDB_C025935 | PGDB_AS000370 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | PTK2 | - | Mino | CN116239566A | PGDB_A065735 | PGDB_C025946 | PGDB_AS000370 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | Mino | CN116239566A | PGDB_A067036 | PGDB_C025950 | PGDB_AS000370 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | PTK2 | - | Mino | CN116239566A | PGDB_A070619 | PGDB_C019619 | PGDB_AS000370 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | Mino | CN116239566A | PGDB_A076308 | PGDB_C025948 | PGDB_AS000370 | View |