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CNC(=O)c1ccccc1Nc1cc(Nc2cc(C)c(C3CCN(Cc4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC(C)C)ncc1C(F)(F)F| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CAL-62 | CN116239566A | PGDB_A007313 | PGDB_C019620 | PGDB_AS000002 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | PTK2 | - | VCaP | CN116239566A | PGDB_A007856 | PGDB_C019620 | PGDB_AS000495 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | Hep3B2.7-1 | CN116239566A | PGDB_A040628 | PGDB_C019620 | PGDB_AS001369 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CCRF-CEM | CN116239566A | PGDB_A044568 | PGDB_C019620 | PGDB_AS000686 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | SW620 | CN116239566A | PGDB_A050607 | PGDB_C019620 | PGDB_AS001904 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CCRF-CEM | CN116239566A | PGDB_A055258 | PGDB_C019620 | PGDB_AS000686 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | VCaP | CN116239566A | PGDB_A060530 | PGDB_C019620 | PGDB_AS000495 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | MM.1S | CN116239566A | PGDB_A076352 | PGDB_C019620 | PGDB_AS000943 | View |