Assay
PGDB_AS000002
System: cell_basedCell line: CAL-62
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CAL-62 | CN116239566A | PGDB_A007313 | PGDB_C019620 | PGDB_AS000002 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | CAL-62 | CN116239566A | PGDB_A007522 | PGDB_C019625 | PGDB_AS000002 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CAL-62 | CN116239566A | PGDB_A012156 | PGDB_C019628 | PGDB_AS000002 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CAL-62 | CN116239566A | PGDB_A014464 | PGDB_C019627 | PGDB_AS000002 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CAL-62 | CN116239566A | PGDB_A024428 | PGDB_C019629 | PGDB_AS000002 | View | |
| IC50 | - | = | 50-100 | nM | - | — | PTK2 | - | CAL-62 | CN116239566A | PGDB_A030586 | PGDB_C019623 | PGDB_AS000002 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CAL-62 | CN116239566A | PGDB_A033927 | PGDB_C019622 | PGDB_AS000002 | View | |
| IC50 | - | = | 50-100 | nM | - | — | PTK2 | - | CAL-62 | CN116239566A | PGDB_A040499 | PGDB_C019626 | PGDB_AS000002 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CAL-62 | CN116239566A | PGDB_A049445 | PGDB_C019624 | PGDB_AS000002 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CAL-62 | CN116239566A | PGDB_A064071 | PGDB_C019621 | PGDB_AS000002 | View |