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CNC(=O)c1ccccc1Nc1cc(Nc2cc(C)c(C3CCN(Cc4ccc5c(c4F)CN(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC(C)C)ncc1C(F)(F)F| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | Hep3B2.7-1 | CN116239566A | PGDB_A037936 | PGDB_C019621 | PGDB_AS001369 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | MGC-803 | CN116239566A | PGDB_A045419 | PGDB_C019621 | PGDB_AS001972 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CCRF-CEM | CN116239566A | PGDB_A052685 | PGDB_C019621 | PGDB_AS000686 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | VCaP | CN116239566A | PGDB_A054848 | PGDB_C019621 | PGDB_AS000495 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | MM.1S | CN116239566A | PGDB_A056491 | PGDB_C019621 | PGDB_AS000943 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CAL-62 | CN116239566A | PGDB_A064071 | PGDB_C019621 | PGDB_AS000002 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | SW620 | CN116239566A | PGDB_A065218 | PGDB_C019621 | PGDB_AS001904 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CCRF-CEM | CN116239566A | PGDB_A065456 | PGDB_C019621 | PGDB_AS000686 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | VCaP | CN116239566A | PGDB_A075328 | PGDB_C019621 | PGDB_AS000495 | View |