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CNC(=O)c1ccccc1Nc1cc(Nc2cc(C)c(N3CCN(Cc4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)cc2OC(C)C)ncc1C(F)(F)F| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | SW620 | CN116239566A | PGDB_A011183 | PGDB_C019629 | PGDB_AS001904 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | CAL-62 | CN116239566A | PGDB_A024428 | PGDB_C019629 | PGDB_AS000002 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | VCaP | CN116239566A | PGDB_A037607 | PGDB_C019629 | PGDB_AS000495 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | MGC-803 | CN116239566A | PGDB_A058695 | PGDB_C019629 | PGDB_AS001972 | View |