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Cc1cc(Nc2ncc(Cl)c(Nc3ccccc3S(=O)(=O)C(C)C)n2)c(OC(C)C)cc1C1CCN(Cc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 100-500 | nM | - | — | ALK | - | NCI-H2228 | CN116239566A | PGDB_A009822 | PGDB_C025908 | PGDB_AS002251 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | PC-9 | CN116239566A | PGDB_A021240 | PGDB_C025908 | PGDB_AS000139 | View | |
| IC50 | - | < | 50 | nM | - | — | ALK | - | SR | CN116239566A | PGDB_A027096 | PGDB_C025908 | PGDB_AS001815 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | MDA-MB-231 | CN116239566A | PGDB_A047651 | PGDB_C025908 | PGDB_AS000594 | View |