Assay
PGDB_AS002251
System: cell_basedCell line: NCI-H2228
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 100-500 | nM | - | — | ALK | - | NCI-H2228 | CN116239566A | PGDB_A009822 | PGDB_C025908 | PGDB_AS002251 | View | |
| IC50 | - | = | 100-500 | nM | - | — | ALK | - | NCI-H2228 | CN116239566A | PGDB_A023157 | PGDB_C019610 | PGDB_AS002251 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | ALK | - | NCI-H2228 | CN116239566A | PGDB_A029506 | PGDB_C025916 | PGDB_AS002251 | View | |
| IC50 | - | = | 50-100 | nM | - | — | ALK | - | NCI-H2228 | CN116239566A | PGDB_A031477 | PGDB_C016074 | PGDB_AS002251 | View | |
| IC50 | - | = | 100-500 | nM | - | — | ALK | - | NCI-H2228 | CN116239566A | PGDB_A036389 | PGDB_C019613 | PGDB_AS002251 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | ALK | - | NCI-H2228 | CN116239566A | PGDB_A067046 | PGDB_C025912 | PGDB_AS002251 | View |