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CC(C)(O)c1cc2nc(C3CCN(Cc4ccc5c(c4F)CN(C4CCC(=O)NC4=O)C5=O)CC3)oc2cc1NC(=O)c1cccc(C(F)(F)F)n1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 50-100 | nM | - | — | IRAK4 | - | MM.1R | CN116239566A | PGDB_A017397 | PGDB_C025959 | PGDB_AS000191 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | Jurkat | CN116239566A | PGDB_A052177 | PGDB_C025959 | PGDB_AS000478 | View | |
| IC50 | - | = | 100-500 | nM | - | — | IRAK4 | - | CAL-62 | CN116239566A | PGDB_A056727 | PGDB_C025959 | PGDB_AS000175 | View |