Assay
PGDB_AS000191
System: cell_basedCell line: MM.1R
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | MM.1R | CN116239566A | PGDB_A009575 | PGDB_C025965 | PGDB_AS000191 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | MM.1R | CN116239566A | PGDB_A013771 | PGDB_C025960 | PGDB_AS000191 | View | |
| IC50 | - | = | 50-100 | nM | - | — | IRAK4 | - | MM.1R | CN116239566A | PGDB_A017397 | PGDB_C025959 | PGDB_AS000191 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | IRAK4 | - | MM.1R | CN116239566A | PGDB_A031820 | PGDB_C025966 | PGDB_AS000191 | View | |
| IC50 | - | = | 100-500 | nM | - | — | IRAK4 | - | MM.1R | CN116239566A | PGDB_A034204 | PGDB_C025963 | PGDB_AS000191 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | MM.1R | CN116239566A | PGDB_A052888 | PGDB_C025954 | PGDB_AS000191 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | MM.1R | CN116239566A | PGDB_A076180 | PGDB_C025953 | PGDB_AS000191 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | MM.1R | CN116239566A | PGDB_A076471 | PGDB_C019639 | PGDB_AS000191 | View |