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Compound
PGDB_C029749
6 activity records1 related patents
2D structure
C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CC6(COc7ccc(N8CCC(=O)NC8=O)cc7C6)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.24 | nM | - | — | AR | - | VCaP | WO2026061104A1 | PGDB_A000140 | PGDB_C029749 | PGDB_AS000481 | View |
| % Degradation | - | = | 8 | % | 5 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A005849 | PGDB_C029749 | PGDB_AS001354 | View |
| % Degradation | - | = | 6 | % | 10 nM | - | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A006299 | PGDB_C029749 | PGDB_AS002463 | View |
| % Degradation | - | = | 19 | % | 50 nM | - | AR | - | VCaP | WO2026061104A1 | PGDB_A078859 | PGDB_C029749 | PGDB_AS001838 | View |
| IC50 | - | = | 0.68 | nM | - | — | AR | - | LNCaPFGC | WO2026061104A1 | PGDB_A078900 | PGDB_C029749 | PGDB_AS000195 | View |