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SIMM · NJU
Assay
PGDB_AS002463
System: cell_based
Target: AR
Cell line: LNCaPFGC
Assay context summary
Assay context
418 activity records
Assay family
% Degradation
System
cell_based
Readout
% Degradation
Target
AR
E3
Not specified
Cell line
LNCaPFGC
Organism
Homo sapiens
Technology
Western_blot
Detection target
protein_degradation
Activity compounds and values
Activity records
418 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
% Degradation
-
=
48
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000040
PGDB_C029743
PGDB_AS002463
View
% Degradation
-
=
18
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000042
PGDB_C030080
PGDB_AS002463
View
% Degradation
-
=
81
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000070
PGDB_C029979
PGDB_AS002463
View
% Degradation
-
=
33
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000087
PGDB_C029897
PGDB_AS002463
View
% Degradation
-
=
55
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000089
PGDB_C030021
PGDB_AS002463
View
% Degradation
-
=
34
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000144
PGDB_C029828
PGDB_AS002463
View
% Degradation
-
=
20
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000146
PGDB_C029940
PGDB_AS002463
View
% Degradation
-
=
12
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000153
PGDB_C029765
PGDB_AS002463
View
% Degradation
-
=
79
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000154
PGDB_C030107
PGDB_AS002463
View
% Degradation
-
=
83
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000261
PGDB_C029807
PGDB_AS002463
View
% Degradation
-
=
86
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000295
PGDB_C029802
PGDB_AS002463
View
% Degradation
-
=
75
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000298
PGDB_C029729
PGDB_AS002463
View
% Degradation
-
=
9
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000299
PGDB_C029941
PGDB_AS002463
View
% Degradation
-
=
59
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000432
PGDB_C030066
PGDB_AS002463
View
% Degradation
-
=
59
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000451
PGDB_C030122
PGDB_AS002463
View
% Degradation
-
=
58
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000516
PGDB_C030008
PGDB_AS002463
View
% Degradation
-
=
65
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000549
PGDB_C029812
PGDB_AS002463
View
% Degradation
-
=
85
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000553
PGDB_C029830
PGDB_AS002463
View
% Degradation
-
=
79
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000565
PGDB_C030081
PGDB_AS002463
View
% Degradation
-
=
56
%
10 nM
-
AR
-
LNCaPFGC
WO2026061104A1
PGDB_A000625
PGDB_C029997
PGDB_AS002463
View