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Nc1nnc(-c2cc(F)ccc2O)cc1N1CC2CCC(C1)N2c1ccc(N2CCN(Cc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4)CC2)cc1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 200-500 | nM | - | — | - | - | H838 | WO2026061475A1 | PGDB_A000616 | PGDB_C030352 | PGDB_AS000282 | View | |
| IC50 | - | = | 500-700 | nM | - | — | - | - | CFPAC-1 | WO2026061475A1 | PGDB_A001872 | PGDB_C030352 | PGDB_AS000179 | View | |
| IC50 | - | = | 5-10 | nM | - | — | - | - | H2126 | WO2026061475A1 | PGDB_A002733 | PGDB_C030352 | PGDB_AS001417 | View | |
| IC50 | - | = | 700-900 | nM | - | — | - | - | A549 | WO2026061475A1 | PGDB_A002940 | PGDB_C030352 | PGDB_AS000757 | View | |
| IC50 | - | = | 200-500 | nM | - | — | - | - | A375 | WO2026061475A1 | PGDB_A078074 | PGDB_C030352 | PGDB_AS002441 | View | |
| IC50 | - | = | 1-5 | nM | - | — | - | - | H1944 | WO2026061475A1 | PGDB_A080593 | PGDB_C030352 | PGDB_AS001924 | View |